Recent advances in the study on capsaicinoids and capsinoidsLUO, Xiu-Ju; JUN PENG; LI, Yuan-Jian et al.European journal of pharmacology. 2011, Vol 650, Num 1, pp 1-7, issn 0014-2999, 7 p.Article

Vanilloid receptor TRPV1 antagonists as the next generation of painkillers. Are we putting the cart before the horse?SZALLASI, Arpad; APPENDINO, Giovanni.Journal of medicinal chemistry (Print). 2004, Vol 47, Num 11, pp 2717-2723, issn 0022-2623, 7 p.Article

Analgesic potential of TRPV1 antagonistsKYM, Philip R; KORT, Michael E; HUTCHINS, Charles W et al.Biochemical pharmacology. 2009, Vol 78, Num 3, pp 211-216, issn 0006-2952, 6 p.Article

ANANDAMIDE AND THE VANILLOID RECEPTOR (TRPV1)TOTH, Attila; BLUMBERG, Peter M; BOCZAN, Judit et al.Vitamins and hormones. 2009, Vol 81, pp 389-419, issn 0083-6729, 31 p.Article

Discovery of novel pyrrolopyridazine scaffolds as transient receptor potential vanilloid (TRPV1) antagonistsDORANGE, Ismet; FORSBLOM, Rickard; MACSARI, Istvan et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 22, pp 6888-6895, issn 0960-894X, 8 p.Article

Structure-activity relationships of vanilloid receptor agonists for arteriolar TRPV1CZIKORA, A; LIZANECZ, E; EDES, I et al.British journal of pharmacology. 2012, Vol 165, Num 6, pp 1801-1812, issn 0007-1188, 12 p.Article

The functions of TRPA1 and TRPV1: moving away from sensory nervesFERNANDES, E. S; FERNANDES, M. A; KEEBLE, J. E et al.British journal of pharmacology. 2012, Vol 166, Num 2, pp 510-521, issn 0007-1188, 12 p.Article

The role of transient receptor potential vanilloid 1 in mechanical and chemical visceral hyperalgesia following experimental colitisMIRANDA, A; NORDSTROM, E; MANNEM, A et al.Neuroscience. 2007, Vol 148, Num 4, pp 1021-1032, issn 0306-4522, 12 p.Article

Clinical development of TRPV1 antagonists : targeting a pivotal point in the pain pathwayGUNTHORPE, Martin J; CHIZH, Boris A.Drug discovery today. 2009, Vol 14, Num 1-2, pp 56-67, issn 1359-6446, 12 p.Article

Characterization of 2-(2,6-dichloro-benzyl)-thiazolo[5,4-d] pyrimidin-7-yl]-(4-trifluoromethyl-phenyl)-amine (JNJ-39729209) as a novel TRPV1 antagonistMAHER, Michael P; BHATTACHARYA, Anindya; YI LIU et al.European journal of pharmacology. 2011, Vol 663, Num 1-3, pp 40-50, issn 0014-2999, 11 p.Article

LASSBio-881: an N-acylhydrazone transient receptor potential vanilloid subfamily type 1 antagonist orally effective against the hypernociception induced by capsaicin or partial sciatic ligationTRIBUTINO, J. L. M; SANTOS, M. L. H; MIRANDA, A. L. P et al.British journal of pharmacology. 2010, Vol 159, Num 8, pp 1716-1723, issn 0007-1188, 8 p.Article

Vanilloid receptor TRPVI is not activated by vanilloids applied intracellularlyVYKLICKY, Ladislav; LYFENKO, Alla; KUFFLER, Damien P et al.Neuroreport (Oxford). 2003, Vol 14, Num 7, pp 1061-1065, issn 0959-4965, 5 p.Article

TRPV3 is a temperature-sensitive vanilloid receptor-like proteinSMITH, G. D; GUNTHORPE, M. J; EGERTON, J et al.Nature (London). 2002, Vol 418, Num 6894, pp 186-190, issn 0028-0836Article

C-fibers, but not the transient potential receptor vanilloid 1 (TRPV1), play a role in experimental allergic airway inflammationROGERIO, Alexandre P; ANDRADE, Edinéia L; CALIXTO, João B et al.European journal of pharmacology. 2011, Vol 662, Num 1-3, pp 55-62, issn 0014-2999, 8 p.Article

Involvement of the transient receptor potential vanilloid 1 (TRPV1) in the development of acute visceral hyperalgesia during colorectal distension in ratsRAVNEFJORD, Anna; BRUSBERG, Mikael; DAIWU KANG et al.European journal of pharmacology. 2009, Vol 611, Num 1-3, pp 85-91, issn 0014-2999, 7 p.Article

Binding of [³H]A-778317 to native transient receptor potential vanilloid-1 (TRPV1) channels in rat dorsal root ganglia and spinal cordBIANCHI, Bruce R; EL KOUHEN, Rachid; JUN CHEN et al.European journal of pharmacology. 2010, Vol 633, Num 1-3, pp 15-23, issn 0014-2999, 9 p.Article

Visceral hypersensitivity induced by activation of transient receptor potential vanilloid type 1 is mediated through the serotonin pathway in rat colonQIN, Hong-Yan; LUO, Jia-Lie; QI, Sheng-Da et al.European journal of pharmacology. 2010, Vol 647, Num 1-3, pp 75-83, issn 0014-2999, 9 p.Article

The effects of a TRPV1 antagonist, SB-705498, in the treatment of seasonal allergic rhinitisBAREILLE, Philippe; MURDOCH, Robert D; DENYER, Jane et al.International journal of clinical pharmacology and therapeutics. 2013, Vol 51, Num 7, pp 576-584, issn 0946-1965, 9 p.Article

The SAR analysis of TRPV1 agonists with the α-methylated B-regionCHO, Yongsung; MYEONG SEOP KIM; HO SHIN KIM et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 16, pp 5227-5231, issn 0960-894X, 5 p.Article

Pungency of TRPV1 agonists is directly correlated with kinetics of receptor activation and lipophilicityURSU, Daniel; KNOPP, Kelly; BEATTIE, Ruth E et al.European journal of pharmacology. 2010, Vol 641, Num 2-3, pp 114-122, issn 0014-2999, 9 p.Article

Rapid disassembly of dynamic microtubules upon activation of the capsaicin receptor TRPV1GOSWAMI, C; DREGER, M; OTTO, H et al.Journal of neurochemistry. 2006, Vol 96, Num 1, pp 254-266, issn 0022-3042, 13 p.Article

Capsazepine, a vanilloid receptor antagonist, inhibits allergen-induced tracheal contractionVAN DEN WORM, Edwin; DE VRIES, Annick; NIJKAMP, Frans P et al.European journal of pharmacology. 2005, Vol 518, Num 1, pp 77-78, issn 0014-2999, 2 p.Article

N-isoquinolin-5-yl-N'-aralkyl-urea and -amide antagonists of human vanilloid receptor 1JETTER, Michele C; YOUNGMAN, Mark A; MCNALLY, James J et al.Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 12, pp 3053-3056, issn 0960-894X, 4 p.Article

Potent and orally efficacious benzothiazole amides as TRPV1 antagonistsBESIDSKI, Yevgeni; BROWN, William; JONES, Paul et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 19, pp 6205-6211, issn 0960-894X, 7 p.Article

Rat detrusor overactivity induced by chronic spinalization can be abolished by a transient receptor potential vanilloid 1 (TRPV1) antagonistSANTOS-SILVA, André; CHARRUA, Ana; CRUZ, Célia D et al.Autonomic neuroscience : basic & clinical. 2012, Vol 166, Num 1-2, pp 35-38, issn 1566-0702, 4 p.Article